Evaluation of the Therapeutic Efficacy of the Newly Formulated Drug “Novostron” as an Experimental Basis for Clinical Trials

Nailya Ibragimova, Aisulu Kabdraisova, Marina Lyu, Zhanar Iskakbayeva, Arkadiy Krasnoshtanov, Yuliya Tin, Sakhipov Yermek, Seitzhan Turganbay, Roza Karzhaubayeva, Aleksander Ivanovich Ilin, Amirkan Azembayev, Serzhan Mombekov and Saki Raheem 2025. Evaluation of the Therapeutic Efficacy of the Newly Formulated Drug “Novostron” as an Experimental Basis for Clinical Trials. ACS Omega. 10 (33), pp. 36946-36959. https://doi.org/10.1021/acsomega.4c11017

TitleEvaluation of the Therapeutic Efficacy of the Newly Formulated Drug “Novostron” as an Experimental Basis for Clinical Trials
TypeJournal article
AuthorsNailya Ibragimova, Aisulu Kabdraisova, Marina Lyu, Zhanar Iskakbayeva, Arkadiy Krasnoshtanov, Yuliya Tin, Sakhipov Yermek, Seitzhan Turganbay, Roza Karzhaubayeva, Aleksander Ivanovich Ilin, Amirkan Azembayev, Serzhan Mombekov and Saki Raheem
Abstract

Chronic wound infections driven by multidrug-resistant (MDR) bacteria continue to challenge modern medicine. This study introduces “Novostron”, an innovative topical iodine-based formulation incorporating dextrin and metal halides designed to overcome the limitations of existing antiseptics, such as volatility and cytotoxicity. The complex’s physicochemical properties were analyzed using infrared (IR) and ultraviolet (UV) spectroscopy, alongside thermogravimetric analysis, confirming its stability and robust iodine retention. Stability assessments revealed minimal iodine loss under optimal refrigerated conditions. In a rat skin wound model, the microbial load was significantly reduced to 1.4 ± 0.5 CFU/cm2 within 10 min postapplication, demonstrating rapid antimicrobial action. Wound-healing properties were evaluated on surgically induced wounds in mice, showing accelerated granulation tissue formation and epithelialization within 14 days, supported by histological findings. In infected wound models, combined therapy with “Novostron” and cefazolin enhanced immune responses (IgG and IgM levels), significantly reduced inflammation, and promoted robust tissue regeneration. Additionally, hematological studies revealed decreased leukocytes and thrombocytes, indicating reduced systemic inflammation. These findings suggest the potential of “Novostron” as a therapeutic agent for managing infected and surgical wounds, offering both antimicrobial and wound-healing benefits. However, clinical trials are essential to validate its safety, optimize its application protocol, and establish its efficacy for human use.

JournalACS Omega
Journal citation10 (33), pp. 36946-36959
ISSN2470-1343
Year2025
PublisherAmerican Chemical Society (ACS)
Publisher's version
License
CC BY 4.0
File Access Level
Open (open metadata and files)
Digital Object Identifier (DOI)https://doi.org/10.1021/acsomega.4c11017
Web address (URL)https://pubs.acs.org/doi/10.1021/acsomega.4c11017
Publication dates
Published13 Aug 2025
Supplemental file
File Access Level
Open (open metadata and files)

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